SEROTONIN AGENTS Flashcards
BUSPIRONE
Buspar
5HT1A
Inhibits 5HT release
Buspar
BUSPIRONE
5HT1A
Inhibits 5HT release
SUMATRIPTAN
Imigran
5HT1D/1B
Vasoconstriction
NARATRIPTAN
Amerge
5HT1D/1B
Vasoconstriction
ZOLMITRIPTAN
Zomig
5HT1D/1B
Vasoconstriction
RIZATRIPTAN
Maxalt
5HT1D/1B
Vasoconstriction
FROVATRIPTAN
Frova
5HT1D/1B
Vasoconstriction
ELETRIPTAN
Replax
5HT1D/1B
Vasoconstriction
ALMOTRIPTAN
Axert
5HT1D/1B
Vasoconstriction
Imigran
SUMATRIPTAN
5HT1D/1B
Vasoconstriction
Amerge
NARATRIPTAN
5HT1D/1B
Vasoconstriction
Zomig
ZOLMITRIPTAN
5HT1D/1B
Vasoconstriction
Maxalt
RIZATRIPTAN
5HT1D/1B
Vasoconstriction
Frova
FROVATRIPTAN
5HT1D/1B
Vasoconstriction
Replax
ELETRIPTAN
5HT1D/1B
Vasoconstriction
Axert
ALMOTRIPTAN
5HT1D/1B
Vasoconstriction
ERGOTAMINE
Gynergen
5HT2A
Vasoconstriction (Vasoselective)
Gynergen
ERGOTAMINE
5HT2A
Vasoconstriction (Vasoselective)
ERGONOVINE
ERGOMETRINE
Ergotrate
5HT2A
Uterine constriction (Uteroselective)
METHYLERGONOVINE
METHYLERGOMETRINE
Methergine
5HT2A
Uterine constriction (Uteroselective)
Ergotrate
ERGONOVINE
ERGOMETRINE
5HT2A
Uterine constriction (Uteroselective)
Methergine
METHYLERGONOVINE
METHYLERGOMETRINE
5HT2A
Uterine constriction (Uteroselective)
Lysergic Acid Diethylamide
LSD
Delysid
5HT2A
CNS selective
Delysid
Lysergic Acid Diethylamide
5HT2A
CNS selective
PHENOXYBENZAMINE
Dibenzyline
α-1 & α-2 nonselective receptor antagonist
Vasodilator
Dibenzyline
PHENOXYBENZAMINE
α-1 & α-2 nonselective receptor antagonist
Vasodilator
CYPROHEPTADINE
Periactin
5HT2A Antagonist
CNS for serotonin syndrome (Vasodilator)
Periactin
CYPROHEPTADINE
5HT2A Antagonist
CNS for serotonin syndrome (Vasodilator)
LORCASERIN
Belviq
5HTC
For obesity
Belviq
LORCASERIN
5HTC
For obesity
FLIBANSERIN
Addyi
5HT2A & 5HT1A
For Hypoactive Sexual Desire Disorder (HSDD) in women
Addyi
FLIBANSERIN
5HT2A & 5HT1A
For Hypoactive Sexual Desire Disorder (HSDD) in women
TEGASEROD
WITHDRAWN: Increase Heart attack & Stroke
Zelnorm
5HT4
GIT motility
Zelnorm
WITHDRAWN: Increase Heart attack & Stroke
TEGASEROD
5HT4
GIT motility
CISAPRIDE
WITHDRAWN: Fatal Arrhythmia
Prospulsid
5HT4
GIT motility
Prospulsid
WITHDRAWN: Fatal Arrhythmia
CISAPRIDE
5HT4
GIT motility
ALOSETRON
Lotronex
5HT3 antagonist
Anti-emetic
ONDANSETRON
Zofran
5HT3 antagonist
Anti-emetic
PALONOSETRON
Aloxi
5HT3 antagonist
Anti-emetic
DOLASETRON
Anzemet
5HT3 antagonist
Anti-emetic
GRANISETRON
Kytril
5HT3 antagonist
Anti-emetic
Lotronex
ALOSETRON
5HT3 antagonist
Anti-emetic
Zofran
ONDANSETRON
5HT3 antagonist
Anti-emetic
Aloxi
PALONOSETRON
5HT3 antagonist
Anti-emetic
Anzemet
DOLASETRON
5HT3 antagonist
Anti-emetic
Kytril
GRANISETRON
5HT3 antagonist
Anti-emetic