Redline and Bolded drugs - French Flashcards
Chlorpromazine (*red)
Typical antipsychotic (D2 antagonist)
Haloperidol (*red)
Typical antipsychotic (D2 antagonist)
Clozapine (*red)
Atypical antipsychotic (D2/5HT2 antagonist)
Olanzapine
Atypical antipsychotic (D2/5HT2 antagonist)
Quetiapine (*red)
Atypical antipsychotic (D2/5HT2 antagonist)
Risperidone
Atypical antipsychotic (D2/5HT2 antagonist)
Aripiprazole
Atypical antipsychotic (D2/5HT2 antagonist)
Fluoxetine (*red)
Antidepressant (Prozac®)
Serotonin Specific Reuptake Inhibitor (SSRI)
Paroxetine (*red)
Antidepressant
Serotonin Specific Reuptake Inhibitor (SSRI)
Sertraline
Antidepressant
Serotonin Specific Reuptake Inhibitor (SSRI)
Escitralopram (*red)
Antidepressant
Serotonin Specific Reuptake Inhibitor (SSRI)
Citalopram
Antidepressant
Serotonin Specific Reuptake Inhibitor (SSRI)
Bupropion (*red)
Antidepressant
Norepinephrine Dopamine Reuptake Inhibitor (NDRI)
Wellbutrin, Zyban (smoking cessation)
Venlafaxine (*red)
Antidepressant
Serotonin Norepinephrine Reuptake Inhibitor (SNRI)
Duloxetine
Antidepressant
Serotonin Norepinephrine Reuptake Inhibitor (SNRI)
Trazodone (*red)
Antidepressant
Mixed Serotonin Reuptake Blocker / Receptor Antagonist
Mirtazipine
Antidepressant
Alpha-2 adrenergic antagonist
Amitriptyline (*red)
Antidepressant
Tricyclic antidepressant (NET /SERT reuptake)
Nortriptyline
Antidepressant
Tricyclic antidepressant (NET /SERT reuptake)
Imipramine
Antidepressant
Tricyclic antidepressant (NET /SERT reuptake)
Desipramine
Antidepressant
Tricyclic antidepressant (NET /SERT reuptake)
Clomipramine
Antidepressant
Tricyclic antidepressant (NET /SERT reuptake)
Phenelzine (*red)
Antidepressant
MAOI (Monoamine Oxidase Inhibitor)
Lithium carbonate (*red)
Antimanic agent
Valproate
Antimanic agent
Alprazolam (*red)
Anxiolytic (Xanax)
Benzodiazepine (BDZ) Agonists (GABA-Cl− channel)
Flurazepam (*red)
Anxiolytic
Benzodiazepine (BDZ) Agonists (GABA-Cl− channel)
Contraindications: elderly
Diazepam (*red)
Anxiolytic (Valium)
Benzodiazepine (BDZ) Agonists (GABA-Cl− channel)
Triazolam (*red)
Anxiolytic
Benzodiazepine (BDZ) Agonists (GABA-Cl− channel)
Oxazepam (*red)
Anxiolytic
Benzodiazepine (BDZ) Agonists (GABA-Cl− channel)
Lorazepam (*red)
Anxiolytic
Benzodiazepine (BDZ) Agonists (GABA-Cl− channel)
Midazolam (*red)
Anxiolytic
Benzodiazepine (BDZ) Agonists (GABA-Cl− channel)
Temazepam (*red)
Anxiolytic
Benzodiazepine (BDZ) Agonists (GABA-Cl− channel)
Flumazenil (*red)
BDZ receptor ANTAgonist
Zolpidem (*red)
Sleep aid (Ambien®, Ambien CR)
BDZ agonist, GABAa only (cortex)
Eszopiclone (*red)
Sleep aid (Lunesta)
BDZ agonist, GABAa only (cortex)
Zaleplon (*red)
Sleep aid (Sonata)
BDZ agonist, GABAa only (cortex)
Phenobarbital (*red)
Barbiturates (GABA-Cl− channel)
Ramelteon (*red)
Sleep aid
Melatonin receptor agonist
Buspirone
5HT1A partial agonist
Diphenhydramine (*red)
Sedative (Benadryl)
Buprenorphine (*red)
x
Disulfiram (*red)
Antabuse
Naltrexone (*red)
x
Clonidine (*red)
x
d-Amphetamine (*red)
Stimulant (Adderall)
ADHD
Methylphenidate (*red)
Stimulant (Ritalin)
ADHD
Desflurane
Volatile anesthetic
Enflurane
Volatile anesthetic
Halothane (*red)
Volatile anesthetic
Isoflurane
Volatile anesthetic
Sevoflurane
Volatile anesthetic
Dantrolene sodium
Malignant hyperthermia (Halothane antidote)
Valproic acid
Antiseizure
contraindicated in pregnancy
Levetiracetam (*red)
Antiseizure
Mechanism unknown (Ca channel) 1st line tx of generalized tonic-clonic
Lamotrigine
Antiseizure
1st line for partial or generalized seizures
Suppress VSSC and VSCC (decreased glu release)
Ethosuximide (*red)
Antiseizure (absence seizures)
GI upset
Valproate (Valproic acid) (*red)
Broad spectrum antiseizure. Blocks T-type Ca channels
TERATOGENIC EFFECTS
GI upset
Hepatic failure
Phenytoin (*red)
Anti-seizure medication (Grand mal aka tonic clonic)
GINGIVAL HYPERPLASIA
CLASSIC INDUCER of P450
Carbamazepine (*red)
Anti-seizure medication (Grand mal aka tonic clonic)
Anti-manic agent
AGRANULOCYTOSIS
Hepatotoxicity
Also a P450 inducer
Lamotrigine
Anti-seizure medication (Grand mal aka tonic clonic) [Lamictal]
Effects on VSSCs (suppress repetitive APs) and VSCCs ( Glu release)
Levetiracetam (*red)
Anti-seizure medication (Grand mal aka tonic clonic)
Phenobarbital (*red)
Anti seizure (Broad spectrum)
Divalproex
Broad spectrum antiseizure (Depakote)
Ethosuximide
Anti-seuzure [Absence (Petit Mal)]
These two drugs cause agranulocytosis
Carbamazepine
Clozapine
Neuroleptic Malignant Synrome is caused by ___?
Atypical antipsychotics