Quick Cards for Targets of Targeted Drugs Flashcards

1
Q

Crizotinib

A

ALK, HGFR

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2
Q

Dasatinib

A

SRC, Bcr-abl, c-KIT, PDGFR

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3
Q

Erlotinib

A

EGFR

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4
Q

Gefitinib

A

EGFR

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5
Q

Imatinib

A

Bcr-abl, c-KIT, and PDGFR

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6
Q

Lapatinib

A

EGFR, HER2

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7
Q

Nilotinib

A

Bcr-abl, c-KIT, and PDGFR

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8
Q

Pazopanib

A

VEGFR, PDGFR, c-KIT

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9
Q

Sorafenib

A

BRAF, VEGFR, PDGFR

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10
Q

Sunitinib

A

VEGFR, PDGFR, c-KIT

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11
Q

Vemurafenib

A

BRAF

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12
Q

Bevacizumab

A

VEGF

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13
Q

Cetuximab

A

EGFR

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14
Q

Panitumumab

A

EGFR

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15
Q

Rituximab

A

CD20

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16
Q

Trastuzumab

A

HER-2

17
Q

Ipilimumab

A

CTLA-4

18
Q

Ofatumumab

A

CD20

19
Q

Bortezomib

A

26-S proteasome inhibitor

20
Q

Vismodegib

A

Hedgehog pathway inhibitor