Midterm Drugs Flashcards

1
Q

Captopril

A

ACE inhibitor

“-pril”

Vasodilator

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2
Q

Enalapril

A

ACE inhibitor

“-pril”

Vasodilator

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3
Q

tPA (plasminogen actvtr)

A

activator of plasminogen

Thrombolytic

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4
Q

Clopidogrel

A

ADP receptor antagonist

Irreversible

“-gel” or “-grel”

Antiplatelet

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5
Q

Prasurgel

A

ADP receptor antagonist

Irreversible

“-gel” or “-grel”

Antiplatelet

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6
Q

Ticagrelor

A

ADP receptor antagonist

Reversible

“-gel” or “-grel”

Antiplatelet

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7
Q

Dobutamine

A

Adrenergic agonist

“A2,B1”

Adrenergic

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8
Q

Dopamine

A

Adrenergic agonist

D1

Adrenergic

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9
Q

Epinephrine

A

Adrenergic agonist

“A1,A2,B1,B2”

Adrenergic

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10
Q

Isoproterenol

A

Adrenergic agonist

“B1,B2”

Adrenergic

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11
Q

Norepinephrine

A

Adrenergic agonist

“A1,A2,B1”

Adrenergic

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12
Q

Eplerenone

A

Aldosterone receptor antagonist

“-one”

Vasodilator

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13
Q

Spironolactone

A

Aldosterone receptor antagonist

“-one”

Vasodilator

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14
Q

Brimonidine

A

Alpha agonist

“A1,A2”

“-ine”

Adrenergic

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15
Q

Clonidine

A

Alpha agonist

A2

“-ine”

Vasodilator

Adrenergic

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16
Q

Midodrine

A

Alpha agonist

non-selective

“-ine”

Adrenergic

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17
Q

Oxymetazoline

A

Alpha agonist

“A1,A2”

“-ine”

Adrenergic

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18
Q

Phenylephrine

A

Alpha agonist

non-selective

“-ine”

Adrenergic

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19
Q

Pazosin

A

Alpha blocker

A1

“-sin”

Vasodilator

Adrenergic

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20
Q

Phenoxybenzamine

A

Alpha blocker

non-selective

Adrenergic

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21
Q

Phentolamine

A

Alpha blocker

non-selective

Vasodilator

Adrenergic

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22
Q

Tamsulosin

A

Alpha blocker

A1

“-sin”

Adrenergic

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23
Q

Terazosin

A

Alpha blocker

A1

“-sin”

Adrenergic

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24
Q

Fondaparinux

A

Antithrombin catalyst

Inhibition of Factor Xa

Anticoagulant

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25
Heparin (UFH)
Antithrombin catalyst inhibition of thrombin Anticoagulant
26
LMWH
Antithrombin catalyst Inhibition of Factor Xa Anticoagulant
27
Losarten
ARB Vasodilator
28
Hydralazine
Arteriolar dilator Vasodilator
29
Albuterol
Beta agonist B2 "-lol" Adrenergic
30
Atenolol
Beta blocker B1 "-lol" Vasodilator Antianginal Adrenergic Antiarrhythmic
31
Esmolol
Beta blocker "-lol" Vasodilator Adrenergic
32
Metaprolol
Beta blocker B1 "-lol" Adrenergic Antiarrhythmic
33
Pindolol
Beta blocker "B1,B2" "-lol" Adrenergic
34
Propanolol
Beta blocker non-selective "-lol" Vasodilator, Antianginal, Adrenergic, Antiarrhythmic
35
Sotalol
Beta blocker non-selective "-lol" Vasodilator, Antianginal, Adrenergic, Antiarrhythmic
36
Cholestyramine
Bile Acid Binding Resin Hypolipidemic
37
Colesevelam
Bile Acid Binding Resin Hypolipidemic
38
Colestipol
Bile Acid Binding Resin Hypolipidemic
39
Ranolazine
Block late sodium current Antianginal
40
Diltiazem
Calcium blocker benzothiazepine Antianginal Antiarrhythmic
41
Amlodipine
Calcium blocker (dihydropridine) " "-pine" Vasodilator
42
Clevidipine
Calcium blocker (dihydropridine) " "-pine" Vasodilator
43
Nicardipine
Calcium blocker (dihydropridine) "-pine" Vasodilator
44
Nifedipine
Calcium blocker (dihydropridine) "-pine" Vasodilator Antianginal
45
Nimodipine
Calcium blocker (dihydropridine) "-pine" Antianginal
46
Verapamil
Calcium blocker (non-dihydropyridine) Vasodilator Antianginal Antiarrhythmic
47
Ezetimibe
Cholesterol absorption inhibitor Hypolipidemic
48
Aspirin
COX Inhibitor Antiplatelet
49
Fenoldopam
Dopamine agonist D1 Vasodilator Adrenergic
50
Procainamide
Fast sodium blocker (Ia) active state Antiarrhythmic
51
Fenofibrate
Fibrate PPAR(alpha) agonist Hypolipidemic
52
Eptifibatide
GPIIa/IIIb inhibitor derivative snake venom Antiplatelet
53
Tirofiban
GPIIa/IIIb inhibitor "synthetic, non-peptide" Antiplatelet
54
Atorvastatin
HMG-CoA Reductase Inhibitor "-statin" Hypolipidemic
55
Lovastatin
HMG-CoA Reductase Inhibitor "-statin" Hypolipidemic
56
Pravastatin
HMG-CoA Reductase Inhibitor "-statin" Hypolipidemic
57
Rosuvastatin
HMG-CoA Reductase Inhibitor "-statin" Hypolipidemic
58
Simvastatin
HMG-CoA Reductase Inhibitor "-statin" Hypolipidemic
59
Dipyridamole
Inhibits cGMP/cAMP PDE Inc cGMP/cAMP Antiplatelet
60
Amiodarone
K+ blocker Antiarrhythmic
61
Bretylium
K+ blocker Antiarrhythmic
62
Ibutilide
K+ blocker Antiarrhythmic
63
Adenosine
K+ channel opener Antiarrhythmic
64
Minoxidil
K+ channel opener Vasodilator
65
Abciximab
MAB against platelet GPIIb/IIIa Antiplatelet
66
Carvedilol
Mixed blocker "A1,B1,B2" "ilol"" or ""alol" Vasodilator Adrenergic Antiarrhythmic
67
Labetalol
Mixed blocker "A1,B1,B2" "ilol"" or ""alol" Vasodilator Adrenergic
68
Bethanechol
Muscarinic agonist Cholinergic
69
Muscarine
Muscarinic agonist Cholinergic
70
Pilocarpine
Muscarinic agonist Cholinergic Anticholinergic
71
Atropine
Muscarinic antagonist Anticholinergic
72
Benztropine
Muscarinic antagonist Anticholinergic
73
Iptratropium
Muscarinic antagonist Anticholinergic
74
Oxybutynin
Muscarinic antagonist Anticholinergic
75
Propantheline
Muscarinic antagonist Anticholinergic
76
Scopolamine
Muscarinic antagonist Anticholinergic
77
Tiotropium
Muscarinic antagonist Anticholinergic
78
Tolterodine
Muscarinic antagonist Anticholinergic
79
Digoxin
Na-K ATPase blocker Antiarrhythmic Positive Inotropic
80
Guanethidine
NE blocker/depletion Adrenergic
81
Amphetamine
NE displacement Adrenergic
82
Ephedrine
NE displacement Adrenergic
83
Nicotine
Nicotinic agonist Cholinergic
84
Varenicline
Nicotinic agonist Partial (a4b2) Cholinergic
85
Hexamethonium (C6)
Nicotinic antagonist Anticholinergic
86
Trimethaphan
Nicotinic antagonist Anticholinergic
87
Isosorbide dinitrate
NO donor "-nitrate" or "Nitro-" Antianginal
88
Isosorbide-5-mononitrate
NO donor "-nitrate" or "Nitro-" Antianginal
89
Nitroglycerin
NO donor "-nitrate" or "Nitro-" Vasodilator Antianginal
90
Sodium Nitroprusside
NO donor "-nitrate" or "Nitro-" Vasodilator
91
Apixiban
Oral direct Factor Xa inhibitor Anticoagulant
92
Rivaroxaban
Oral direct Factor Xa inhibitor Anticoagulant
93
Dabigatran
Oral direct thrombin inhibitor Anticoagulant
94
Inamrinone
PDE inhibitor Vasodilator Positive Inotropic
95
Cilostazol
PDE-3 inhibitor Inc cAMP Antiplatelet
96
Milrinone
PDE-3 inhibitor Vasodilator Positive Inotropic
97
Laropiprant
PGD2 antagonist (used w/ niacin) Hypolipidemic
98
Streptokinase
Plasmin enhancers Derived from Strep Thrombolytic
99
Urokinase
Plasmin enhancers Derived from kidneys Thrombolytic
100
Aliskiren
Renin inhibitor Vasodilator
101
Bivalirudin
reversible, direct thrombin inhibitors synth deriv of leeches Anticoagulant
102
Lepirudin
reversible, direct thrombin inhibitors synth deriv of leeches Anticoagulant
103
Argatroban
small molec. Inhibitor thrombin Anticoagulant
104
Flecainide
Sodium blocker (Ic) Antiarrhythmic
105
Lidocaine
Very fast sodium blocker (Ib) active/inactive state Antiarrhythmic
106
Warfarin
Vit K-epoxide reductase inhibitor 4-hydroxycoumarins Anticoagulant
107
Niacin
VLDL secretion inhibitor Hypolipidemic