Medication Names Flashcards
Naloxone
Opioid antidote
Rapidly reverses respiratory depression due to pure opioid intoxication
Naltrexone
Prevents euphoric effects of opioids & alcohol, so patients can quit
Must be opioid free for 7-10 days otherwise can precipitate opioid withdrawal
Hepatotoxic & causes liver dysfunction
Methylnaltrexone, Naloxegol, Naldemedine
Opioid antagonists for clients that have constipation with long term opioid use
Are not reversal agents & do not precipitate withdrawal
Adenosine
Anti-arrhythmic used to treat SVT & Wolff parkinson white syndrome
Can cause brief asystole
Tamsulosin, Terazosin, Doxazosin, Prazosin
Alpha-1 Adrenergic Receptors
Treats hypertension & benign prostatic hyperplasia
Valsartan, Irbesartan, Losartan, Telmisartan
Angiotensin II Receptor Blockers (ARBs)
Causes vasodilation, excretion of sodium & water
Treats hypertension, heart failure, MI, diabetic nephropathy, chronic kidney disease
Captopril, Enalapril, Lisinopril, Ramipril
Angiotensin-Converting Enzyme Inhibitors (ACE)
Causes vasodilation & inhibits breakdown of bradykinin
Treats hypertension, heart failure, MI, chronic kidney disease, diabetic nephropathy
Can cause dry cough, hyperkalemia
Warfarin
Anticoagulant
Takes 5-7 days for full effect
Teratogenic
Rivaroxaban, Apixaban
Anticoagulant - Direct Factor Xa Inhibitors
Rapid effect
Renal & hepatic impairment
Dabigatran, Argatroban, Desirudin, Bivalirudin
Anticoagulant - Direct Thrombin Inhibitors
Does not require lab monitoring
Heparin
Activates antithrombin –> does not influence clot that already exists
Antidote = protamine sulfate
Enoxaparin, Dalteparin
Low molecular weight heparin
not aPPT monitoring required
Clopidogrel, Prasugrel, Ticagrelor
Antiplatelet
Treats angina, MI, stent placement, ischemic stroke, peripheral artery disease
Antidote = abciximab, eptifibatide, tirofiban
Metoprolol, Atenolol
Cardio-selective B1 Receptor Blocker (Beta Blocker)
Acts on heart to reduce heart rate, decrease myocardial oxygen demand & decrease cardiac workload
Propranolol, Timolol
Nonselective B1 & B2 receptor blockers (Beta Blockers)
Reduce bronchoconstriction in lungs & reduce HR
Carvedilol, Labetalol
Block alpha, B1 & B2 receptors (Beta Blockers)
Vasodilation in peripheral vasculature, decrease HR & BP
Colesevelam, Cholestyramine, Colestipol
Bile acid sequestrants
Prevents reabsorption & increase excretion if bile acids
Reduce LDL; hypercholesterolemia
Calcium
Antidote for magnesium toxicity
Amlodipine, Nifedipine, Nicardipine, Felodipine
Calcium Channel Blockers - Dihydropyridines
Promote vascular smooth muscle relaxation to decrease BP & systemic vascular resistance
Treat hypertension, chronic stable angina, Raynaud phenomenon
Verapamil & Diltiazem
Calcium Channel Blockers - Non-Dihydropyridines
Decrease HR & increase peripheral vasodilation
Treats angina, a-fib, a-flutter, SVT
Digoxin & Digitoxin
Cardiac Glycosides
Decreases HR & helps heart pump more forcefully at slower rate
Treats heart failure & A-fib
Interacts with diuretics, aminoglycosides & amiodarone (hypokalemia & nephrotoxic)
Lovastatin, Simvastatin, Pravastatin, Atorvastatin, Rosuvastatin
HMG-CoA Reductase Inhibitor
Reduces LDL
Can cause hepatotoxicity
Fenofibrate, Gemfibrozil
Fibrates
Triglyceride lowering
Nitroglycerin
Vasodilation, reduces preload & cardiac oxygen demand
Treats angina
Alteplase, Tenecteplase, Reteplase
Thrombolytics
Dissolves clot, restores blood flow & perfusion
Treats MI, ischemic stroke, massive PE, clotted catheters
Phytonadione
Vitamin K supplement
Methimazole & Propylthiouracil
Anti-thyroid (Thioamides)
Block production of T3 & T4
Takes 3-12 weeks to control symptoms of hyperthyroidism
Causes hepatotoxicity & agranulocytosis
Lispro, Aspart & Glulisine Insulin
Rapid acting
Onset 15 min, peak 1-2 hours, lasting 3-4 hours
NPH insulin
Intermediate acting
onset 1-2 hours, speak 4- 10 hours, duration 14-20 hours
Given 2x daily for basal coverage
Glargine, Degludec, Detemir insulin
Long acting
onset 3-4 hours, no peak, duration 24 hours
Metformin
Biguanides - Oral antidiabetic
Decreases production production in liver & sensitizes insulin receptors in tissues
Do not stimulate pancreas to release more insulin
Alogliptin, Linagliptin, Saxagliptin, Sitagliptin
Dipeptidyl Peptidase 4 inhibitors - Oral antidiabetics
Increase glucose dependent insulin release
Nateglinide, Repaglinide
Meglitinides - Oral antidiabetics
Stimulate release of insulin
Canagliflozin, Dapagliflozin, Empagliflozin
Sodium-Glucose Cotransporter 2 (SGLT-2) Inhibitors - Oral Antidiabetics
Promotes glucose excretion
Glipizide, Glyburide, Glimepiride
Sulfonylureas - Oral Antidiabetics
Stimulate increased release of insulin
Pioglitazone, Rosiglitazone
Thiazolidinedione - Oral Antidiabetics
Increase insulin receptor sensitivity
Levothyroxine
Treatment of hypothyroidism