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IT 1 (MedChem) > IT 1 (MedChem) > Flashcards

IT 1 (MedChem) Flashcards

1
Q

2-phenylethylamine (PEA)

A

base structure for adrenergic agonists

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2
Q

norepinephrine

A

nonselective adrenergic agonist
B1 preference
low affinity for B2

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3
Q

epinephrine

A

nonselective agonist
B > a preference

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4
Q

isoproterenol

A

PEA derivative
B selective (bulky R1) agonist

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5
Q

methyl-DOPA

A

PEA derivative
prodrug for a-methyl norepinephrine
a2 selective agonist
antihypertensive

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6
Q

metaproterenol

A

PEA derivative
B2 selective (bulky R1) agonist

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7
Q

phenylephrine

A

PEA derivative
a selective agonist
for hypotension and nasal congestion

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8
Q

L-DOPS

A

PEA derivative
nonselective adrenergic agonist
prodrug for norepinephrine
for orthostatic hypotension

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9
Q

dipivefrin

A

PEA derivative
nonselective B agonist
prodrug for epinephrine

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10
Q

lisdexamphetamine

A

PEA derivative
prodrug for dexamphetamine
nonselective adrenergic agonist
for ADHD

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11
Q

ephedrine/pseudoephedrine

A

PEA derivative
nonselective adrenergic agonist
nasal decongestant

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12
Q

midodrine

A

PEA derivative
prodrug
a1 selective agonist
for orthostatic hypotension

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13
Q

isoproterenol

A

template 1 analog
nonselective B agonist
for heart block

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14
Q

albuterol, terbutaline

A

template 1 derivative
B2 selective agonist
for asthma (short-acting)

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15
Q

salmeterol, vilanterol, formoterol

A

template 1 analog
B2 selective agonist
for asthma (long-acting)

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16
Q

indacaterol, olodaterol

A

template 1 analog
B2 selective agonist
for asthma (ultra long-acting)

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17
Q

cocaine, amphetamines

A

PEA derivative
nonselective, indirect adrenergic agonist

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18
Q

bupropion

A

PEA derivative
nonselective, indirect adrenergic agonist
for depression and smoking cessation

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19
Q

oxymetazoline

A

template 2 analog
a1 selective agonist
for nasal congestion

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20
Q

clonidine

A

template 2 analog
a2 selective agonist
INDIRECT a1 antagonist

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21
Q

guanfacine

A

noncyclic template 2 analog
a2 selective agonist
ADHD

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22
Q

prazosin

A

a1 selective antagonist
for hypertension

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23
Q

terazosin, doxazosin

A

a1 selective antagonist
for hypertension + BPH

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24
Q

alfuzosin, tamsulosin, silodosin

A

a1 selective antagonist
for BPH

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25
Q

yohimbine

A

a2 selective antagonist
for vet med

26
Q

reserpine

A

indirect adrenergic antagonist
VMAT inhibitor

27
Q

deutetrabenazine

A

first FDA approved deuterated drug
for Huntington’s disease

28
Q

valbenazine

A

prodrug for tardive dyskinesia

29
Q

propranolol

A

aryloxypropanolamine template
1st generation
nonselective B antagonist

30
Q

atenolol, metoprolol

A

aryloxypropanolamine template
2nd generation
B1 selective antagonist

31
Q

carvedilol, labetalol

A

aryloxypropanolamine template
3rd generation
mixed adrenergic antagonist (B1, B2, a1)

32
Q

timolol

A

no aryloxypropanolamine template
nonselective B antagonist
for glaucoma

33
Q

acetylcholine

A

nonselective cholinergic agonist
miosis

34
Q

miochol E

A

acetylcholine salt form
nonselective cholinergic agonist
for miosis

35
Q

methacholine

A

acetylcholine derivative
nonselective cholinergic agonist
M preference
for asthma test

36
Q

carbachol

A

acetylcholine derivative
nonselective cholinergic agonist
N preference
for miosis

37
Q

bethanechol

A

acetylcholine derivative
nonselective cholinergic agonist
M preference
for urinary retention

38
Q

tetra methyl ammonium

A

N selective agonist

39
Q

tetra ethyl ammonium

A

N selective antagonist

40
Q

hexa methonium

A

N ganglion blocker

41
Q

deca methonium

A

N depolarizing neuromuscular blocker
cholinergic agonist
for muscle relaxation

42
Q

succinylcholine

A

acetylcholine dimer
N depolarizing neuromuscular blocker
cholinergic agonist
for muscle relaxation

43
Q

phenyl trimethyl ammonium

A

N selective agonist

44
Q

choline

A

N selective agonist
choline reuptake inhibitor

45
Q

nicotine

A

N agonist
for smoking cessation

46
Q

cytisine

A

N partial agonist
for smoking cessation

47
Q

imidacloprid

A

N agonist
for insecticide

48
Q

bupropion

A

N channel blocker
for depression + smoking cessation

49
Q

mecamylamine

A

N channel blocker
for hypertension

50
Q

tubocurarine, malouetine

A

natural product
nondepolarizing skeletal neuromuscular blocker
N cholinergic antagonist

51
Q

muscarine

A

natural product
M selective agonist

52
Q

pilocarpine

A

natural product
M selective agonist
for glaucoma, xerostomia, Sjogren’s

53
Q

cevimeline

A

M selective agonist
for Sjogren’s

54
Q

atropine

A

M selective antagonist
for pre-op, cardiovascular, muscarine toxicity, mydriasis

55
Q

homatropine

A

M selective antagonist
for ophthalmic

56
Q

ipratropium

A

M selective antagonist
for bronchodilation

57
Q

tiotropium

A

M selective antagonist
for bronchospasm

58
Q

trospium

A

M selective antagonist
for urinary incontinence

59
Q

scopolamine

A

M selective antagonist
for nausea, ophthalmic, antispastic

60
Q

methscopolamine

A

M selective antagonist
for nasal decongestion, anticholinergic

IT 1 (MedChem) (1 decks)

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