Hypertension Formulary Test Flashcards
Amlodipine (Norvasc) Dosages
2.5mg, 10mg
Amlodipine (Norvasc) SE/Monitoring
Reflex tachycardia, flushing, dizziness, headaches, peripheral edema, gingival hyperplasia
Increased risk of angina/MI in pts w/ obstructive coronary disease
DRUG INTERACTIONS: grapefruit juice, CYP3A4 enzyme inducers/inhibitors
Amlodipine (Norvasc) Drug Class
DHP CCB
Atenolol (Tenormin) Dosages
25mg, 50mg, 100mg
Atenolol (Tenormin) SE/Monitoring
Dizziness, fatigue, weakness
Monitor for swelling, passing out, or slow heartbeat
Atenolol (Tenormin) Drug Class
BBs
Benazepril (Lotensin) Dosages
5mg, 10mg, 20mg, 40mg
Benazepril (Lotensin) SE/Monitoring
Angioedema, cough (up to 20%), hyperkalemia, acute renal failure
NOT FOR pregnant people
Benazepril (Lotensin) Drug Class
ACEi
Clonidine (Catapres) Dosages
PO - 0.1mg, 0.2mg
Transdermal - 0.1-0.3mg/day
Clonidine (Catapres) SE/Monitoring
CNS depression, dizziness, fatigue, anticholinergic effects, bradycardia, reflex tachycardia, fluid retention
Clonidine (Catapres) Drug Class
Central Alpha-2 Agonists
Carvedilol (Coreg) Dosages
6.25/dose, 50mg (BID)
Carvedilol (Coreg) SE/Monitoring
Bronchospasm, bradycardia, fatigue, exercise intolerance, depression
CI: 2nd/3rd deg heart block, decompensated HF, Post-MI, severe bradycardia, sick sinus syndrome
Carvedilol (Coreg) Drug Class
Mixed Alpha/Beta
Enalapril (Vasotec) Dosages
5mg, 40mg
Enalapril (Vasotec) SE/Monitoring
Angioedema, cough (up to 20%), hyperkalemia, acute renal failure
NOT FOR pregnant people
Enalapril (Vasotec) Drug Class
ACEi
Hydrochlorothiazide (Microzide) Dosages
12.5mg, 50mg
Hydrochlorothiazide (Microzide) SE/Monitoring
Hyperkalemia, hypomagnesemia, hypercalcemia, hyperuricemia, hyperglycemia, hyperlipidemia, sexual dysfunction, increase in TG/cholesterol
DRUG INTERACTIONS: lithium toxicity
CI: sulfa allergy, anuria
Dose in the AM
Hydrochlorothiazide (Microzide) Drug Class
Thiazide Diuretic
Labetalol (Trandate) Dosages
100mg/dose, 800mg (BID)
Labetalol (Trandate) SE/Monitoring
Bronchospasm, bradycardia, fatigue, exercise intolerance, depression
CI: 2nd/3rd deg heart block, decompensated HF, Post-MI, severe bradycardia, sick sinus syndrome
Labetalol (Trandate) Drug Class
Mixed Alpha/Beta
Lisinopril (Zetril) Dosages
10mg, 40mg
Lisinopril (Zetril) Drug Class
ACEi
Lisinopril (Zetril) SE/Monitoring
Angioedema, cough (up to 20%), hyperkalemia, acute renal failure
NOT FOR pregnant people
Losartan (Cozaar) Dosages
50mg, 100mg
Losartan (Cozaar) SE/Monitoring
Angioedema, hyperkalemia, acute renal failure
DO NOT give to pregnant people
Losartan (Cozaar) Drug Class
ARBs
Metoprolol succinate (Toprol XL) Dosages
25mg, 400mg
Metoprolol succinate (Toprol XL) SE/Monitoring
Bronchospasm, bradycardia, fatigue, exercise intolerance, depression
CI: 2nd/3rd deg heart block, decompensated HF, Post-MI, severe bradycardia, sick sinus syndrome
Metoprolol succinate (Toprol XL) Drug Class
Cardioselective BBs
Metoprolol tartrate (Lopressor) Dosages
50mg/dose, 450mg BID
Metoprolol tartrate (Lopressor) SE/Monitoring
Bronchospasm, bradycardia, fatigue, exercise intolerance, depression
CI: 2nd/3rd deg heart block, decompensated HF, Post-MI, severe bradycardia, sick sinus syndrome
Metoprolol tartrate (Lopressor) Drug Class
Cardioselective BBs
Nifedipine (Procardia) Dosages
30mg, 120mg
Nifedipine (Procardia) SE/Monitoring
Reflex tachycardia, flushing, dizziness, headaches, peripheral edema, gingival hyperplasia
Increased risk of angina/MI in pts w/ obstructive coronary disease
DRUG INTERACTIONS: grapefruit juice, CYP3A4 enzyme inducers/inhibitors
Nifedipine (Procardia) Drug Class
DHP CCBs
Spironolactone (Aldactone) Dosages
12.5mg, 100mg
Spironolactone (Aldactone) SE/Monitoring
Hyperkalemia, hyponatremia, gynecomastia
DRUG INTERACTIONS: ACEi/ARBs/Renin inhibitors/NSAIDs - increased risk of hyperkalemia
CI: potassium sparing diuretics
Spironolactone (Aldactone) Drug Class
Aldosterone Antagonist
Valsartan (Diovan) Dosages
80mg, 320mg
Valsartan (Diovan) SE/Monitoring
Angioedema, hyperkalemia, acute renal failure
DO NOT give to pregnant people
Valsartan (Diovan) Drug Class
ARBs
Hyzaar (losartan + HCTZ) Dosages
50mg/12.5mg; 100mg/25mg
Lotrel (amlodipine + benazepril) Dosages
2.5mg/10; 10mg/40mg
Maxzide (HCTZ + triamterene) Dosages
25mg/37.5mg; 50mg/75mg
Zestoretic (lisinopril + HCTZ) Dosages
10mg/12.5mg; 80mg/50mg
Monitoring for ACEi/ARBs
BUN/SCr, K
Monitoring for CCBs
HR (non-DHP)
Monitoring for Aldosterone Antagonists
BUN/SCr, K
Monitoring for other diuretics
BUN/SCr, electrolytes (K, Mg, Na), uric acid (thiazides)
Monitoring for BBs
HR