Guess the drug Flashcards
Acetylcholine
Carbachol
Pilocarpine
Bethanechol
Cholinergic direct acting
Galantamine Donepezil Rivastgmine Neostigmine Physostigmine Edrophonium Pyridostigmine
Cholinergic indirect acting
Used to treat Myasthenia Gravis:
Galantamine Donepezil Rivastgmine Neostigmine Physostigmine Edrophonium Pyridostigmine
Edrophonium
Treats anticholinergic poisoning:
Galantamine Donepezil Rivastgmine Neostigmine Physostigmine Edrophonium Pyridostigmine
Physostigmine
Reverses effects of anaesthetics:
Galantamine Donepezil Rivastgmine Neostigmine Physostigmine Edrophonium Pyridostigmine
Neostigmine, Pyridostigmine
Alzheimers disease:
Galantamine Donepezil Rivastgmine Neostigmine Physostigmine Edrophonium Pyridostigmine
Galantamine
Donepezil
Rivastgmine
Atropine Scopolamine Ipratropium Tiotropium Oxybutynin Trospium
Anticholinergic agonists
Toilet:
Atropine Scopolamine Ipratropium Tiotropium Oxybutynin Trospium
Oxybutynin
Trospium
Vomitting, motion sickness:
Atropine Scopolamine Ipratropium Tiotropium Oxybutynin Trospium
Scopolamine
Stimulates GI tract, trachychardia, mydriasis, blocks glands:
Atropine Scopolamine Ipratropium Tiotropium Oxybutynin Trospium
Atropine
Bronchodilation, which one lasts longer?
Which one treats runny noses?
Atropine Scopolamine Ipratropium Tiotropium Oxybutynin Trospium
Ipratropium, Tiotropium
Tiotropium lasts longer than ipratropium.
Ipratropium is also used as nasal sprays to treat runny noses
Which one releases the Laudanosine poision?
Cisatracurium Vecuronium Pancuronium Atracurium Rocuronium
Non- depolarising neuromuscular blockers
Atracurium
Succinylcholine
Depolarising neuromuscular blocker
Nicotine
Ganglionic blocker
Prazosin Silodoozin Phentolamine Doxazosin Tamsulosin Phenaxybenzamine Terazosin Alfuzosin
Alpha blockers
Non- selective alpha blockers?
Prazosin Silodoozin Phentolamine Doxazosin Tamsulosin Phenaxybenzamine Terazosin Alfuzosin
Phentolamine
Phenaxybenzamine
Irreversible agonist vs reversible?
Phentolamine
Phenaxybenzamine
• Phenaxybenzamine is an irreversible antagonist
- Phentolamine is a reversible antagonist
Selective alpha blockers that lower blood pressure?
Prazosin Silodoozin Phentolamine Doxazosin Tamsulosin Phenaxybenzamine Terazosin Alfuzosin
Prazosin, Doxazosin, Terazosin
Selective alpha blockers that help with enlarged prostates?
Prazosin Silodoozin Phentolamine Doxazosin Tamsulosin Phenaxybenzamine Terazosin Alfuzosin
Tasulosin, Alfuzosin and Silodozin
Which ones don’t belong as beta blockers?
Carvedilol Carbachol Sotalol Nadolol Propranolol Esmolol Formoterol Metaprolol Betaxolol Nebivolol Pindolol Salmeterol Acebutolol Albuterol Timolol Sotalol Atenolol Bisoprolol Labetalol
Formoterol
Albuterol
Salmeterol
Carbachol
Propranolol Pindolol Nadolol Sotalol Timolol
First generation non-selective beta blockers
Bisoprolol Atenolol Esmolol Metaprolol Acebutolol
Second generation B1 selective beta blockers
Carvedilol
Labetalol
Third generation non- selective B and A1 beta blockers
Betaxolol
Nebivolol
Third generation non- selective B1 beta blockers
Mirabegron Chlonadine Salmeterol Terbutaline Phenylephrine Albuterol Formoterol Dobutamine Oxymetazoline
Selective adrenergic agonists
A1 selective
Eyes:
Runny nose:
Mirabegron Chlonadine Salmeterol Terbutaline Phenylephrine Albuterol Formoterol Dobutamine Oxymetazoline
Oxymetazoline
Phenylephrine
B3 selective
Toilet:
Mirabegron Chlonadine Salmeterol Terbutaline Phenylephrine Albuterol Formoterol Dobutamine Oxymetazoline
Mirabegron
A2 selective
Blood pressure, withdrawal symptoms:
Mirabegron Chlonadine Salmeterol Terbutaline Phenylephrine Albuterol Formoterol Dobutamine Oxymetazoline
Chlonadine
B1 selective
Increases heart rate:
Mirabegron Chlonadine Salmeterol Terbutaline Phenylephrine Albuterol Formoterol Dobutamine Oxymetazoline
Dobutamine
B2 selective
Bronchodilators
Mirabegron Chlonadine Salmeterol Terbutaline Phenylephrine Albuterol Formoterol Dobutamine Oxymetazoline
Albuterol and Terbutaline
Salmeterol and Formoterol
Epinephrine
Norepinephrine
Dopamine
Non- selective direct acting adrenergic agonists
Cocaine and Amphetamine
Indirect acting adrenergic agonists
Ephedrine
Pseudoephedrine
Mixed action adrenergic agonists