GENERAL Flashcards

1
Q

Lugares donde se encuentra M1

A

estómago, células parietales gástricas

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2
Q

Lugares donde se encuentra M2

A

corazón, células cardíacas y musculares lisas

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3
Q

Lugares donde se encuentra M3

A

músculo liso, glándulas exócrinas, vejiga.

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4
Q

Receptores muscarínicos que activan la vía Gq, por ende generan respuestas mediadas por CALCIO

A

M1, M3, M5

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5
Q

Receptores muscarínicos que se acoplan a proteína G, Gi Gq para inhibir la adenilato cíclala y regular conductos irónicos específicos

A

M2, M4

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6
Q

Ésteres de colina

A
Metacolina
Acetilcolina
Betanecol
Carbacol
*MABC*
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7
Q

Alcaloides naturales

A

Pilocarpina

Cevimelina

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8
Q

Que familias comprenden los Anticolinesterásicos

A

Inhibidores reversibles
Organofosforados
Carbamiladores

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9
Q

Inhibidores reversibles

A

Tacrina
Edrofonio
Donepezilo
TED

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10
Q

Organofosforados

A

Ecotiofato

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11
Q

Carbamoiladores

A
Fisostigmina
Neostigmina
Rivastigmina
Galantamina
Piridostigmina
Ambenonio
Praliboximina y Obidoximina
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