General Flashcards
Phase 2 …glucuronic acid ?
(🧑⚕️MAC)
Aspirin …morphine….chloramphenicol
Phase 2…Acetic acid (acetylation)?
☄️hip☄️
Isoniazid…hydralazine…procainamide
Phase 2 methylation?
Noradrenaline
Phase2 glycine?
Aspirin
Phase 2 sulfation?
Steroids
Basic drugs ?
Ephidrine….amphetamine
Acidic drugs,?
Aspirin ….barbiturate
Increase rate of gastric empyting ?
Metoclopramide
Decrease rate of gastric empyting ?
Atropine
1- Rapid disintegration?
2- slow disintegration,?
1- paracetamol
2-digoxin
Hepatic first pass?
Pass through liver and distructed via enzymes….(mlpnn)
Morphine …nitroglycrine…lidocaine…propranolol…natural sex hormone
Hepatic enzymes inducers
Phenobarbitone
Phenytoin
Carbamazepine
Rifampicin
Androgen
Tobacco smoke
hepatic enzymes inhibitors specific
Cimetidine
Ciprofloxacin
Chloramphenicol
Erythromycin
Estrogen
Valproic acid
Hepatic enzymes inhibitors non-specific?
hepatotoxic drugs &drugs decreasing hepatic blood flow
as propranolol & cimetidine
Cause absent limbs (phocomelia)
thalidomide
Cardiac septal defect
Aspirin
Cleft palate
Phenytoin
Hepatotoxicity
halothane and paracetamol
Nephrotoxicity
NSAID and aminoglycosides
Neurotoxicity 8 nerve
Streptomycin
Drugs for Alzehimer’s disease?
Galantamine
Rivastigmine
Donepezil
Must be injected very rapidly IV?
Thiopental
Diazoxide
(Because they are highly bound to plasma protein)
Drug not suitable for males as it produces infertility?
……………
كلوربرومازين
Chlorpromazine
Iatro genic disease,? Drug induced diseases?
Salicylate and corticosteroids cause peptic ulcer
Phenothiazine and antisychotics cause parkinsonism