Exam 1 Drugs Flashcards
Plaquenil
hydroxychloroquine
Non-biologic DMARD
T-lymphocyte suppression
Arava
leflunomide
Non-biologic DMARD
Pyrimidine synthase inhibitor
Rheumatrex
methotrexate
Non-biologic DMARD
Dihydrofolate reductase inhibitor
Azulfidine
sulfasalazine
Non-biologic DMARD
Inhibits cytokine secretion
Orencia
abatacept
Biologic DMARD
Inhibits T-cell activation - blocks CD80/86 on APC
Kineret
anakinra
Biologic DMARD
Inhibits IL-1 receptor antagonist
Rituxan
rituximab
Biologic DMARD
Induces B-cell apoptosis - CD20 antibody; binds to CD20 on B cells
Actemra
tocilizumab
Biologic DMARD
Inhibits IL-6
Kevzara
sarilumab
Biologic DMARD
Inhibits IL-6
Humira
adalimumab
DMARD
Binds TNF-a
Cimzia
certolizumab
DMARD
Binds TNF-a
Enbrel
etanercept
DMARD
Binds TNF-a
Simponi
golimumab
DMARD
Binds TNF-a
Remicade
infliximab
DMARD
Binds TNF-a
Xeljanz
tofacitinib
DMARD
Selective JAK inhibitor
Olumiant
baricitinib
DMARD
Selective JAK inhibitor
Rinvoq
upadacitnib
DMARD
Selective JAK inhibitor