estrogens, serms, and progestins Flashcards
natural steroidal estrogens
estradiol, estradiol valerate
synthetic steroidal estrogens
ethinyl estradiol and mestranol
nonsteroidal compounds with estrogenic activity
diethylstilbestol, bisphenol A, and genistein
dosing of ethinyl estradiol for OC
20-35 mcg/day
dosing for premarin for MHT
0.625mg/day
conversion of 0.625mg of CE to ethinyl estradiol
5-10 mcg
drugs used for hot flashes and sweating
estrogen, provera(if estrogen contraindicated), duavee(combines CE with bazedoxifene)
tamoxifen citrate
soltamax, SERM drug
raloxifene
evista, SERM drug
toremifene
fareston (SERM)
clomiphene citrate
clomid (SERM)
fulvestrant
faslodex (Antiestrogen)
ribociclib
kisqali (antiestrogen)
anastrozole
arimidex (nonsteroidal aromatase inhibitor)
letrozole
femara (nonsteroidal aromatase inhibitor)
exemestane
aromasin (steroidal aromatase inhibitor)
1st generation progestins
estranes (nortestosterone and norethindrone)
2nd and 3rd generation progestins
gonanes (norgestrel and norgestimate)
4th generation progestin
drospirenone
which drugs are pregnanes
progesterone and medroxyprogesterone
progesterone drugs
prempro and premphase (contains medroxyprogesterone acetate and CE)
mifepristone
mifeprex (anti-progestin)
misoprostol
cytotec (for ulcers)
notable synthetic progesterones in CHC
levonorgestrel and drospirenone (slynd)
yaz
drospirenone/ethinyl estradiol (OC)
mini pills
progestin only (OC)
post-coital pills
Levonorgestrel (plan B)
myfembree
relugolix, estradiol, and norethindrone acetate) to reduce heavy menstrual bleeding associated with uterine fibroids