Enzyme inducers and inhibitors Flashcards
For each of the drugs, state whether it is an inducer or an inhibitor
Mnemonic for remembering enzyme inducers?
BS CRAP GPS
Mnemonic for remembering enzyme inhibitors?
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Enzyme inducer or inhibitor:
Sodium Valproate
Inhibitor
Enzyme inducer or inhibitor:
St John’s Wort
Inducers
Enzyme inducer or inhibitor:
Carbamazepine
Inducer
Enzyme inducer or inhibitor:
Isoniazid
Inhibitor
Enzyme inducer or inhibitor:
Phenytoin
Inducer
Enzyme inducer or inhibitor:
Alcohol (chronic use)
Inducer
Enzyme inducer or inhibitor:
Erythromycin (and other macrolides)
Inhibitor
Enzyme inducer or inhibitor:
Rifampicin
Inducer
Enzyme inducer or inhibitor:
Omeprazole
Inhibitor
Enzyme inducer or inhibitor:
Alcohol (non-chronic use/binge drinking)
Inhibitor
Enzyme inducer or inhibitor:
Phenobarbital
Inducer
Enzyme inducer or inhibitor:
Cimetidine
Inhibitor
Enzyme inducer or inhibitor:
Fluconazole
Inhibitor
Enzyme inducer or inhibitor:
Griseofulvin
Inducer
Enzyme inducer or inhibitor:
Metronidazole
Inhibitor
Enzyme inducer or inhibitor:
Sulfonylureas
Inducer
Enzyme inducer or inhibitor:
Sulfonamides
Inhibitors
Enzyme inducer or inhibitor:
Chloramphenicol
Inhibitor
Enzyme inducer or inhibitor:
Ketoconazole
Inhibitor
Enzyme inducer or inhibitor:
Ciprofloxacin
Inhibitor
Enzyme inducer or inhibitor:
Barbiturates
Inducer
Enzyme inducer or inhibitor:
Grapefruit juice
Inhibitor