Dyslipidemia Drug Formulary Flashcards
Statins
atorvastatin
rosuvastatin
simvastatin
pravastatin
lovastatin
pitavastatin
fluvastatin
Atorvastatin brand name
Lipitor
Atorvastatin dosing
5 mg, 10 mg, 20 mg, 40 mg, 80 mg
Rosuvastatin brand
crestor
Rosuvastatin dosing
5 mg, 10 mg, 20 mg, 40 mg
Atorvastatin adverse effects and monitoring parameters
muscle toxicity: myopathy, rhabdomyolysis
watch for unusual muscle pain and darkened urine
fatigue
muscle injury: myalgias, myositis, rhabdomyolysis
Rosuvastatin adverse effects and monitoring parameters
muscle toxicity: myopathy, rhabdomyolysis
watch for unusual muscle pain and darkened urine
fatigue
muscle injury: myalgias, myositis, rhabdomyolysis
Simvastatin brand
zocor
Simvastatin dosing
10 mg, 20 mg, 40 mg, 80 mg
Simvastatin adverse effects and monitoring parameters
muscle toxicity: myopathy, rhabdomyolysis
watch for unusual muscle pain and darkened urine
fatigue
muscle injury: myalgias, myositis, rhabdomyolysis
Pravastatin brand
pravachol
Pravastatin dosing
10 mg, 20 mg, 40 mg, 80 mg
Pravastatin adverse effects and monitoring parameters
muscle toxicity: myopathy, rhabdomyolysis
watch for unusual muscle pain and darkened urine
fatigue
muscle injury: myalgias, myositis, rhabdomyolysis
Lovastatin brand
altoprev
mevacor
Lovastatin dosing
10 mg, 20 mg, 40 mg, 80 mg
Lovastatin adverse effects and monitoring parameters
muscle toxicity: myopathy, rhabdomyolysis
watch for unusual muscle pain and darkened urine
fatigue
muscle injury: myalgias, myositis, rhabdomyolysis
Pitavastatin brand
livalo
Pitavastatin dosing
1 mg, 2 mg, 4 mg
Pitavastatin adverse effects and monitoring parameters
muscle toxicity: myopathy, rhabdomyolysis
watch for unusual muscle pain and darkened urine
fatigue
muscle injury: myalgias, myositis, rhabdomyolysis
Fluvastatin brand
lescol
Fluvastatin dosing
20 mg, 40 mg, 80 mg, XL 80 mg
Fluvastatin adverse effects and monitoring parameters
muscle toxicity: myopathy, rhabdomyolysis
watch for unusual muscle pain and darkened urine
fatigue
muscle injury: myalgias, myositis, rhabdomyolysis
Cholesterol absorption inhibitors
ezetimibe
Ezetimibe brand name
zetia
Ezetimibe dosing
10 mg
Ezetimibe adverse effects and monitoring parameters
fatigue
diarrhea
GI upset
PCSK-9 Inhibitors
evolocumab
alirocumab
Evolocumab brand name
repatha
Evolocumab dosing
140 mg every 2 weeks or 240 mg once a month
Evolocumab adverse effects and monitoring parameters
GI upset
increased LFTs
injection site rxn
myalgia
influenza
Alirocumab brand name
praluent
Alirocumab dosing
every 2 weeks either 75 or 150 mg
Alirocumab adverse effects and monitoring parameters
GI upset
increased LFTs
injection site rxn
myalgia
influenza
Bile acid sequestrants
cholestyramine
colesevelam
colestipol
Cholestyramine brand name
questran
prevalite
Cholestyramine dosing
4 g one or two times a day; increase to 8 to 24 g a day
Cholestyramine adverse effects and monitoring parameters
imparied absorption of fat-soluble vitamins (A, D, E, K)
hypernatremia
hyperchloremia
GI obstruction
Colesevelam brand name
WelChol
Colesevelam dosing
625 mg tab, six tabs a day
Colesevelam adverse effects and monitoring parameters
imparied absorption of fat-soluble vitamins (A, D, E, K)
hypernatremia
hyperchloremia
GI obstruction
Colestipol brand name
colestid
Colestipol dosing
2 to 16 g
Colestipol adverse effects and monitoring parameters
imparied absorption of fat-soluble vitamins (A, D, E, K)
hypernatremia
hyperchloremia
GI obstruction
Fibrates
fenofibrate
gemfibrozil
Fenofibrate brand name
Antara, Fenoglide, Lipofen, Lofibra, TriCor, Triglide
Fenofibrate dosing
TriCor tablet: 48mg, 145mg
Lofibra tablet: 54mg, 160mg
Fenoglide tablet: 40mg, 120mg
Triglide tablet: 160mg
Lipofen capsule: 50mg, 150mg
Fenofibrate adverse effects and monitoring parameters
GI disturbances, rash, myalgia, dizziness
Gemfibrozil brand name
lopid
Gemfibrozil dosing
600 mg tab, twice a day
Gemfibrozil adverse effects and monitoring parameters
GI disturbances, rash, myalgia, dizziness
Omega-3 Fatty Acids
omega-3 fatty acid
icosapent ethyl
Others
niacin
Omega-3 fatty acid brand name
lovaza
Omega-3 fatty acid dosing
lovaza: 2-4 g daily or divided BID
Omega-3 fatty acid adverse effects and monitoring parameters
bad breath, GI symptoms
Icosapent ethyl brand name
vascepa
Icosapent ethyl dosing
2 g BID
Icosapent ethyl adverse effects and monitoring parameters
bad breath, GI symptoms
Niacin brand name
niacor
niaspan
slo-niacin
Niacin dosing
500-2000 mg/day
Niacin adverse effects and monitoring parameters
flushing and itching, tingling of upper body, and headache