Drugs to know Flashcards
Tetrodotoxin
voltage gated sodium channel antagonist
Lidocaine
use-dependent voltage gated sodium channel antagonist
Acetylcholine-nicotine
nicotinic agonist
acetylcholine-muscarine
muscarinic agonist
acetylcholine-physostigmine
acetylcholinesterase antagonist
acetylcholine- D-tubocurare
peripheral nicotinic receptor antagonist
acetylcholine- bungarotoxin
peripheral nicotinic receptor antagonist
acetylcholine- atropine
muscarinic receptor antagonist
dopamine-reserpine
blocks dopamine vesicular transporter
dopamine-amphetamine
blocks dopamine vesicular transporter, blocks catecholamine reuptake
dopamine-cocaine
block catecholamine reuptake
dopamine: L-DOPA
drives dopamine biosynthesis
dopamine-chlorpromazine
D2 antagonist
norepinephrine-isoproterenol
beta 1 agonist
norepinephrine-phenylephrine
alpha 1 agonist
norepinephrine- propanolol
beta 2 antagonist
norepinephrine-yohimbine
alpha 2 antagonist
serotonin fluoxetine (Prozac)
serotonin reuptake inhibitor
serotonin-LSD
5-HT6/7 agonist
serotonin-sumatriptin
5-HT1d agonist
serotonin-clozapine
5-HT7 antagonist
histamine-diphenylhydramine
H1 antagonist
histamine-lorantidine
H1 antagonist
glutamate-AMPA
AMPA agonist
glutamate-CNQX
AMPA antagonist
glutamate-NMDA
NMDA agonist
glutamate-AP-5
competitive NMDA antagonist
glutamate-PCP
non-competitive NMDA antagonist
GABA-benzodiazepines (diazepam)
potentiates GABA signalling
GABA-muscimol
GABAA agonist
GABA-bicuculline
GABAA antagonist
GABA-pentobarbital
potentiates GABA signalling
GABA-baclofen
GABAB agonist
GABA-phaclofem
GABAB antgonist
opiates
opiate receptor agonist
naloxone
opiate antagonist
tetrahydrocannibinol
cannabinoid agonist
caffeine
adenosine receptor antagonist