Drugs, receptors, and mechanisms Flashcards
Doxazosin
a1 antagonist
Pilocarpine
M agonist (direct–ACh analogue)
Epinepherine
a1-B1-B2 agonist
Labetalol
a1-B1-B2 antagonist
Pralidoxime- 2PAM
Chlolinesterase reactivation to treat organophosphate poisoning
Ipratroprium
M antagonist (competitive)
Organophosphate Nerve Gasses
M agonist (indirect–irreversible AChE inhibitor)
Oxybutynin/Tolterodine
M antagonist (competitive)
Pseudoephedrine
a1-B2 agonist
Curare/Atracurium/Rocuronium
Nicotinic muscular AChR blocker (non-depolarizing)
Norepinephrine
a1-B1 agonist
Neostigmine/Pyridostigmine
M agonist (indirect–reversible AChE inhibitor)
Albuterol
B2 agonist
Metoprolol/Atenolol
B1 antagonist
Edrophonium
M agonist (indirect–reversible AChE inhibitor)
Succinylcholine
Depolarizing NM blocker
Propranolol
B1-B2 antagonist
Phenylephrine
a1 agonist
Bethanechol
M agonist (direct--ACh analogue) selective for muscarinic--no effect on nicotinic
Atropine/Scopolamine
M antagonist (competitive)
Dobutamine
B1 agonist