Drugs on Histamine Receptor Subtypes Flashcards
Histaprodifen
Partially Selective Agonist of H1
Amthamine
Partially Selective Agonist of H2
R-α-Methylhistamine
Partially Selective Agonist of H3
Imetit
Partially Selective Agonist of H3 and H4
Immepip
Partially Selective Agonist of H3
Clobenpropit
Partially Selective Agonist of H4
Clozapine
Partially Selective Agonist of H4
Triprolidine
Partially Selective Antagonist of H1
Cetirizine
Partially Selective Antagonist of H1
Tiotidine
Partially Selective Antagonist of H2
Iodophenpropit
Partially Selective Antagonist of H3
Proxyfan
Partially Selective Antagonist of H3
Mepyramine
Partially Inverse Agonist of H1
Cimetidine
Partially Inverse Agonist of H2
Ranitidine
Partially Inverse Agonist of H2
Thioperamide
Partially Inverse Agonist of H3 and H4
Clobenpropit
Partially Inverse Agonist of H3