DRUGS Flashcards
Local Anesthetics types
(Na channel blockers) Esters, Amides, Na channel toxins
LA Amides
Lidocaine, Bupivacaine
LA esters
Cocaine, Procaine
LA Na channel toxins
Saxitoxin, Tetrodotoxin (TTX)
Opioid Analgesics categories
Agonists (mu) Combination with NSAIDs Antidiarrheals Antitussive Mixed Agonist (kappa)/Antagonists (mu) Partial Agonists (mu) Antagonists
Opioid Analgesic Agonists
Morphine, Hydrocodone, Oxycodone, Codeine, Tramadol, Fentanyl
Opioid combo with NSAIDs
codeine-acetamenophen Codeine-aspirin Hydrocodone-acetaminophen Hydrocodone-ibuprofen Oxycodone-acetaminophen
Opioid analgesics: Partial agonists (mu)
Buprenorphine
Opioid Antagonists
Naloxone
Pain Management drug categories
Opioids NSAIDs NMDA receptor antagonists alpha2 agonist Adjuvant analgesics
NSAID categories
Non-selective COX1/COX2 inhibitors
COX-2 selective inhibitors
COX-2 inhibitors (CNS)
Non-selective COX1/2 inhibitors
NSAIDs!
Salicylates: Aspirin, Naproxen, Ibuprofen, Ketoprofen
NMDA receptor antagonist
Ketamine; pain management
Opioid adjuvant analgesics
antidiarrhial, antitussive
Adjuvant analgesics for pain management
antidepressnats, anticonvulsants, Local anesthetic: topical lidocaine
Headache management
Migraine- abortive therapy and prophylactic therapy
Migraine abortive therapy
NSAIDS: ibuprofen, naproxen, acetaminophen
5HT1(D) Agonists: Sumatriptan
Ergot compounds: Dihydroergotamine
Migraine prophylactic therapy
Antihypertensives (beta blockers, Ca channel blocers, ACE inhibitors) Anticonvulsants Ergot alkaloids Antidepressents (SSRIs) Botulinum toxin
Treatment for Wernicke’s encephalopathy
Thiamine
Treatment for Dementia
Cholinesterase inhibitors (Donepezil) NMDA-glutamate antagonists (Memantine)
Stroke Risk Reduction
Antiplatelets (Aspirin CLopidogrel)
Anticoagulants (Warfarin, dabigatran)
Emergency Management Stroke
Thrombolytic therapy: tPA
Emergency Management of subarachnoid hemorrhage
decrease ICP: Mannitol