Drugs 1 Flashcards
alpha1 agonist
Phenylephrine
Tetrahydrozoline
Oxymetazoline
Alpha2 agonist
Clonidine
Xylazine
Non-selective beta agonist
Isoproterenol
beta 1 agonist
Dobutamine
Beta2 agonist
Albuterol
Metaproterenol
Beta3 agonist
Myrbetric
Sympathomimetics
Tyramine
Amphetamines
Catecholamine re-uptake block
Cocaine
Imipramine
Amitryptyline
Mixed acting sympathomimetics
Ephedrine
Pseudoephedrine
Phenylephrine
Blocker of NE release
Guanethidine
Bretylium
Clonidine
Blocker of NE vesicular storage
Reserpine
False transmitter (NE)
Alpha-methyl-DOPA
NE synthesis blockade
Alpha-methyl-p-tyrosine
NE
Disulfiram
Blockade of NE metabolism
Pargyline (MAO)
Moclobemide (MAO)
Tolcapone (COMT)
Irreversible alpha-receptor antagonist
Dibenamine
Phenoxybenzamine
Reversible alpha-receptor antagonist
Phentolamine
Selective alpha1 antagonist
Prazosin
Tamsulosin
Selective alpha2 antagonist
Yohimbine
Non-selective beta antagonist
Propranolol
Pindolol
Timolol
Selective beta1 antagonist
Metoprolol
Selective beta2 antagonist
Butoxamine
Blockage of ACh synthesis/release
Hemicholinium
Vesamicol
Botulinus toxin
Parasympathomimetics
Acetylcholine
MEthacholine
Carbachol
Bethanecol
Naturally occurring parasympathomimetics
Pilocarpine
Arecoline
Muscarine
Muscarinic antagonists
Atropine
Homatropoine
Scopolamine
Propantheline
Tropicamide
Ganglionic nicotinic agonist
Nicotine
Ganglionic nicotinic antagonist
Hexamethonium
Trimethaphan
Reversible AChE antagonist
Edrophonium
Carbamylating AChE antagonist
Physostigmine
Neostigmine
Pyridostigmine
Demecarium
Phosphorylating AChE antagonists
Organophosphates
Diisopropyl fluorophosphoric acid
Treatment for organo-phosphate poisoning
Pralidoxime (2-PAM)
Non-depolarizing competitive antagonists (NM)
D-tubocurarine
Pancuronium
Atracurium
Depolarizing NMJ antagonist
Succinylcholine
Induction of CYP450
Phenobarbitol
Polycyclic aromatic hydrocarbons
Glucocorticoids
Inhibitors of CYP450
Azole family antifungals (ketoconazole)