Drug groups Flashcards
Direct Muscarinic Agonists
Acetylcholine Chloride Methacholine Carbachol Bethanechol Cevimeline Pilocarpine
First Generation ACHE inhibitors
Edrophonium Neostigmine Pyridostigmine Physostigmine Echothiopate
Second Generation ACHE inhibitors
Tacrine
Donepezil
Rivastigmine
Galantamine
Muscarinic Antagonists
Atropine Scopolamine Ipratropium Oxybutynin Tolteridine Darifenacin Solifenacin Glycopyrrolate Benztropine Trihexyphenidyl
Nicotinic Neuronal (NN/N2) receptor agonists and antagonists
Nicotine Varenicline Mecamylamine Trimethaphan Hexamethonium
Non-depolarizing competitive antagonist - neuromuscular junction (NMJ) blocker/SKM relaxing drugs
d-Tubocurarine Atracurium Cis-Atracurium Mivacurium Pancuronium Vecuonium Rocuronium
Depolarizing NMJ antagonist
Succinylcholine
Selective Alpha 1 agonist drugs
Phenylephrine
Midodrine
Selective Alpha 2 agonist drugs
Alpha-Methyldopa Clondine Tizanidine Dexmedetomidine Guanfacine Aproclonidine Brimonidine
Indirect-acting Agonists
Amphetamine-like drugs Tyramine Guanethidine Cocaine Tricyclic antidepressants (TCAs)
Selective Alpha 1 Antagonist drugs (blockers)
Prazosin
Terazosin
Doxazosin
Tamsulosin
Non-selective Mixed (alpha 1 & alpha 2) antagonist drugs
Phentolamine
Phenoxybenzamine
Selective Alpha 2 Antagonist drugs
Yohimbine
Selective Beta 1 Agonist drugs
Dobutamine
Direct Acting Non-selective (beta 1 & beta 2) Agonist drugs
Isoproterenol
Epinephrine (EPI)
Ephedrine
Indirect Acting Beta (beta 1 & beta 2) Agonists
Amphetamine
Tyramine
Tricyclic antidepressants (Amitriptyline, Desipramine, Imipramine, and Nortriptyline)
Selective NE reuptake inhibitors (SNRIs - Atomoxetine)
Cocaine
Non-selective Beta (beta 1 & beta 2) Blockers
Propranolol
Nadolol
Timolol
Pindolol
Cardioselective Beta Blockers (Beta 1 antagonist)
Atenolol Metoprolol Acebutolol Nebivolol Esmolol
A-MANE
ISA (Partial agonists) for beta blockers
Pindolol (beta 1 & 2)
Acebutolol (beta 1 only)
Non-selective Mixed (alpha 1 & beta 1/2) receptor antagonists
Carvedilol
Labetolol
Beta blockers for Glaucoma
Betaxolol
Levobunolol
Timolol
Metipranolol
Selective Beta 2 agonist drugs
Formeterol Terbutalin Salmeterol Albuterol Metaproterenol
ForT SAM
Selective Beta 3 agonist
Mirabegron