Day 1 Flashcards
Edrophonium
Myasthenia gravis diagnosis
Varenecline
Nicotine analog
Smoking cessation
Muscarinic toxicity
CNS stimulation
Nicotinic toxicity
Ganglionic stimulation
Pyridostigmine
Neostigmine
Myasthenia gravis treatment
Inhibit acetylcholinesterase
Rivastigmine
Alzheimer’s
Organophosphate poisoning
Atropine
Pralidoxime
Rivastigmine
Alzheimer’s disease
Inhibit acetylcholinesterase
Memantine
Alzheimer’s disease
NMDA receptor blocker
Succinylcholine
Depolarizing NMB
Hoffman degradation
Atracurium
Atropine toxicity
Hot as a hare Dry as a bone Red as a beet Blind as a bat Mad as a hatter
Contraindications to muscarinic blockers
Infants
AACG
BPH
Scopolamine
Motion sickness
Ipratropium
Muscarinic antagonist
Benztropine
Muscarinic antagonist
Atropine
Muscarinic antagonist
Pralidoxime
Breaks organophosphate bond with cholinesterase
Regenerates acetylcholinesterase
Beta 2 effect on aqueous
Increase
MOA of MAO and COMT
Metabolize (degrade) catecholamines