Cardiovascular drugs - categories only Flashcards
Heparin
anticoagulant
LMWH
anticoagulant
Warfarin
anticoagulant (oral)
Protamine sulfate
anti-heparin
fondaparinux
Anti-10a
Hirudin
HIT-avoidance anti-coagulant
Bivalirudin
HIT-avoidance anti-coagulant
Argatroban
2a inhibitor
AT3 concentrate
anticoagulant
Vitamin K
Warfarin antidote
Recombinant 7a
Warfarin antidote
Fresh frozen plasma
Warfarin antidote
Tirofiban
GPIIa/IIIb inhibitor
Abciximab
GPIIa/IIIb inhibitor
Eptifibamibe
GPIIa/IIIb inhibitor
Zileuton
Leukotriene inhibitor
Monteleukast
Leukotriene inhibitor
Zarirkulast
Leukotriene inhibitor
Clopidogrel
ADP receptor inhibitor
Prasugrel
ADP receptor inhibitor
Ticlopidine
ADP receptor inhibitor
Ticagrelor
ADP receptor inhibitor
Cangrelor
ADP receptor inhibitor
Cilostazol
PDE3 blocker - antiplatelet
Dipyramidol
PDE3 blocker - antiplatelet
Tenecteplase
recombinant t-PA (MI, stroke)
Reteplase
recombinant t-PA (MI, stroke)
Alteplase
recombinant t-PA (MI, stroke)
Streptokinase
recombinant t-PA (PE, MI, stroke)
Urokinase
recombinant t-PA (PE, MI, stroke)
Ancrod
recombinant t-PA (stroke)
Pravustatin
anti-LDL (non CYP)
Rosuvastatin
anti-LDL
Lovastatin
anti-LDL
Fluvastatin
anti-LDL
Simvistatin
anti-LDL
Cholestyramine
anti-LDL (bile acid resin), increases TAG though!
Colestipol
anti-LDL (bile acid resin), increases TAG though!
Colesevalam
anti-LDL (bile acid resin), increases TAG though!
Ezetimebe
Cholesterol absorption inhibitor
Evolocumab
anti-LDL (PCSK9 inhibitor)
Alirocumab
anti-LDL (PCSK9 inhibitor)
Heterozygous for LDLR
Lomitapide
anti-LDL (MTP inhibitor)
Homozygous null LDLR
Mipomerson
anti-LDL (APO-B inhibitor)
Homozygous null LDLR
Niacin
HDL booster
Gemfibrozil
TAG reducer
Fenofibrate
TAG reducer
NO
vasodilator
Nitroprusside
A/V dilator
Hydralazine
vasodilator
Nitroglycerin
vasodilator
Isosorbide dinitrate
vasodilator
Captopril
ACE inhibitor
Lisinopril
ACE inhibitor
Enalapril
ACE inhibitor
Ramipril
ACE inhibitor
Losartan
Angiotensin II receptor blocker (ARB)
Icatibant
Bradykinin receptor blocker
Aprotinin
Kallikrein blocker
Desmopressin
releases endothelial VWF/VIII
Bosentan
Endothelin antagonist
Acetazolamide
CA inhibitor diuretic
Dorzolamide
CA inhibitor diuretic
Methazolamide
CA inhibitor diuretic
Dichlorophenamide
CA inhibitor diuretic
Mannitol
Osmotic diuretic
Furosamide
Loop diuretic
Bumetanide
Loop diuretic
Torsemide
Loop diuretic
Ethacrynic acide
Loop diuretic (for sulfa allergy)
HCTZ
Thiazide diuretic
Chlorothiazide
Thiazide diuretic
Chlorothalidone
Thiazide diuretic
Indapamide
Thiazide diuretic
Metolazone
Thiazide diuretic - for renal failure, non sulfa structure
Spironolactone
K+ sparing diuretic (aldosterone R blocker)
Eplerenone
K+ sparing diuretic (aldosterone R blocker)
Amiloride
K+ sparing diuretic
ENaC block
Triamterene
K+ sparing diuretic
ENaC block
Tolvaptan
AVP receptor blocker
Conivaptan
AVP receptor blocker
Aminocaproic acid
anti-fibrinolytic (pro-clot)
Transexemic acid
anti-fibrinolytic (pro-clot)
Aprotinin (trasylol)
anti-fibrinolytic (pro-clot)
Alpha-2-antiplasmin
anti-fibrinolytic (pro-clot)
PAI-1
anti-fibrinolytic (pro-clot)
13a
anti-fibrinolytic (pro-clot)
Procainamide
Anti-arrhythmic (1A)
Quinidine
Anti-arrhythmic (1A) - cinchonism
Disopyramide
Anti-arrhythmic (1A)
Lidocaine
Anti-arrhythmic (1B)
Mexilitene
Anti-arrhythmic (1B)
Flecainide
Anti-arrhythmic (1C)
Propafenone
Anti-arrhythmic (1C)
Propanalol
nonspecific B-blocker
Antiarrhythmic
Esmolol
B-blocker (short half-life) - antiarrhythmic
Amiodarone
AP prolonger
Anti-arrhythmic (Class III)
Dronedarone
AP prolonger
Anti-arrhythmic (Class III)
Sotalol
AP prolonger (Class III)
Verapimil
CCB: neg ino/chronotrope
Diltiazem
CCB: neg ino/chronotrope
Adenosine
Anti-arrhythmic (temporary flatline…restarts heart)
Nifedipine
CCB
Losartan
ARB
Reserpine
sympatholytic
Methyldopa
sympatholytic
Guanfacine
sympatholytic
Clonidine
sympatholytic
Phenoxybenzamine
non-selective alpha blocker
Prazosin
a1 blocker
Minoxidil
vasodilator
Amlodipine
CCB
Nicarpidine
CCB
Rinolazine
P-Fox blocker to reduce O2 consumption for angina
Ivabradine
I-funny channel blocker (anti-anginal)
Niseritide
venodilator
Nitroglycerin
venodilator
Dobutamine
B1 agonist –> boost CO
Milrinone
PDE-i for acute CHF
Amrinone
PDEI-i for acute CHF
Digitalis
positive inotrope
LCZ696
anti-remodelling