antibiotics vets Flashcards
Penicillins
1. Narrow spectrum penicillins 2. Penicillinase stable penicillins 3. Broad spectrum penicillins 4. Penicillins acting against Pseudomonas spp
Narrow spectrum
penicillins
- benzylpenicillin-Na,K
- benzylpenicillin-procaine
- benzylpenicillin-benzathine
- phenoxymethyl-penicillin
Penicillinase stable
penicillins
- oxacillin
- cloxacillin
- dicloxacillin
- flucloxacillin
Broad spectrum
penicillins
- amoxicillin
2. ampicillin
Penicillins acting against
Pseudomonas spp
- ticarcillin
2. piperacillin
Beta-lactam antibiotics- mode of action
time dependent bactericidal
Beta-lactam antibiotics- mechanism of action
inhibition of cell wall
synthesis
Beta-lactamase-inhibitors
- clavulanic acid
- sulbactam
- tazobactam
Cephalosporins 1st gen.
- cephazoline
- cephapirin
- cefadroxil
- cephalexin
Cephalosporin 2nd gen.
- cefuroxime
Cephalosporin 3rd gen.
- ceftiofur
- cefovecin
- ceftriaxone
- cefotaxime
- ceftazidime
- cefoperazone
Cephalosporin 4th gen.
- cefquinome
Carbapenems
- imipenem
2. meropenem
Beta-lactam antibiotics - Groups
- Penicillins
- Beta-lactamase-inhibitors
- Cephalosporins
- Carbapenems
- Monobactams
Monobactams
- aztreonam
2. tigemonam
Aminoglycosides- mode of action
concentration
dependent
bactericidal
(Except: spectinomycin - bacteriostatic)
Aminoglycosides- mechanism of action
inhibition of protein synthesis (30S
subunit), mistranslation.
Aminoglycosides antibiotics
- streptomycin
- neomycin
- paromomicin
- kanamycin
- gentamicin
- tobramycin
- amikacin
- apramycin
Tetracyclines antibiotics
Short-acting tetracyclines: 1. chlortetrcycline 2. oxytetracycline 3. tetracycline Long-acting tetracyclines: 1. doxycycline 2. minocycline
Tetracyclines- mode of action
bacteriostatic
Tetracyclines- mechanism of action
inhibition of protein synthesis
30S subunit
Macrolides antibiotics
- erythromycin
- azithromycin
- clarithromycin
- spiramycin
- tylosin
- tylvalosin
- tilmicosin
- tulathromycin
- gamithromycin
- tildipirosin
Macrolides- mode of action
bacteriostatic
Macrolides- mechanism of action
inhibition of protein synthesis
50S subunit
Lincosamides antibiotics
- lincomycin
2. clindamycin
Lincosamides- mode of action
bacteriostatic
Lincosamides- mechanism of action
inhibition of protein synthesis
50S subunit
Pleuromutilins antibiotics
- tiamulin
2. valnemulin
Pleuromutilins- mode of action
bacteriostatic
Pleuromutilins- mechanism of action
inhibition of protein synthesis
50S subunit
Phenicols antibiotics
inhibition of protein synthesis
50S subunit
Phenicols- mode of action
bacteriostatic
Phenicols- mechanism of action
inhibition of protein synthesis
50S subunit