ADRENERGIC RECEPTORS Flashcards
α1
Vascular smooth muscle
Vasoconstriction
α1
Radial muscle of iris
Mydriasis
α1
Pilomotor smooth muscle
Contraction
α1
Urinary bladder
Urinary retention
α2
CNS
Inhibition of release catecholamines
α2
Peripheral blood vessels
Vasoconstriction
β1
Heart
Tachycardia
β1
Uterine muscles
Uterine relaxation
β2
Blood vessels
Vasodilation
β1
Liver
Glycogenolysis
β2
Neuromuscular endplates
Hypokalemia
β3
Adipose tissues
Lipolysis
D1
Renal Blood Vessels
Renal vasodilation
D2
GIT
Loss of peristalsis
D2
CNS
Modulation of motor activity perception and behavior
α1
Effector organ/s
- Vascular smooth muscle
- Urinary bladder
- Radial muscle of iris
- Pilomotor smooth muscle
Gq-linked
α2 Pre-synaptic
Effector Organ/s
- CNS
Gi-linked
α2 Post-synaptic
Effector Organ/s
- Peripheral blood vessels
Gq-linked
β1
Effector Organ/s
- Heart
- Juxtaglomerular apparatus
Gs-linked
β2
Effector Organ/s
- Uterine muscles
- Bronchioles
- Blood vessels
- Neuromuscular endplates
- Liver
Gs-linked
β3
Effector Organ/s
- Adipose tissues
Gs-linked
D1
Effector Organ/s
- Renal Blood Vessels
Gs-linked
D2
Effector Organ/s
- GIT
- CNS
Gi-linked