HIV drugs Flashcards
1
Q
elvitegravir (EVG)
A
INSTI
SE: nausea/diarrhea upper resp tract infections, bronchitis back/joint pain UTI drug interactions
2
Q
raltegravir (RAL)
A
INSTI
SE: high creatinine kinase myositis, rhabdomyolosis skin rash hypersensitivity
3
Q
dolutegravir
A
INSTI
4
Q
maraviroc
A
FI
binds ccr5
5
Q
enfuvirtide
A
FI
binds gp41
6
Q
ritonavir (RTV)
A
PI
CYP34A inhibitor
combo w/other PI
induces own metabolism
7
Q
atazanavir
A
PI
8
Q
darunavir
A
PI
9
Q
fosamprenavir
A
PI
10
Q
indinavir
A
PI
11
Q
nelfinavir
A
PI
12
Q
squinavir
A
PI
13
Q
tipranavir
A
PI
14
Q
efavirenzs (EFV)
A
NNRTI
most potent
15
Q
delavirdine
A
NNRTI
16
Q
etravirine
A
NNRTI
17
Q
nevirapine
A
NNRTI
18
Q
rilpivirine
A
NNRTI
19
Q
zidovudine (AZT)
A
NRTI
glucuronidation
20
Q
abacavir (ABC)
A
NRTI
alcohol dehydrogenase
hypersensitivity (test HLAb5701)
21
Q
tenofir disproxil fumarate (TDF)
A
NRTI
22
Q
emtricitabine (FTC)
A
NRTI