Antihistamines, NSAIDs, GI Flashcards
Sodium bicarbonate
Acid-neutralizing agent
Calcium carbonate
Acid-neutralizing agent
TUMS
Magnesium hydroxide/ Aluminum hydroxide
Acid-neutralizing agent
“Tidines”
H2 Histamine Antagonist
Cimetidine
H2 Histamine Antagonist
Ranitidine
H2 Histamine Antagonist
Famotidine
H2 Histamine Antagonist
Nizatidine
H2 Histamine Antagonist
“Prazoles”
PPIs
Omeprazole
PPI
Esomeprazole
PPI
Lansoprazole
PPI
Rabeprazole
PPI
Pantoprazole
PPI
Misoprostol
Cytoprotective agent
Bismuth subsalicylate
Cytoprotective agent
Metoclopramide
Prokinetic agent
Bethanechol
Prokinetic agent
Erythromycin
Prokinetic agent
Dicyclomine
Antispasmotic for IBS
Amitriptyline
Antispasmotic for IBS
Eluxadoline
Antispasmotic for IBS
Glycopyrrolate
Antispasmotic for IBS
Ondasetron
Anti-nausea
Anti-emetic
Serotonin (5HT3)
antagonist
“setrons”
Anti-nausea
Anti-emetic
Serotonin (5HT3) antagonist
Granisetron
Anti-nausea
Anti-emetic
Serotonin (5HT3)
antagonist
Palonosetron
Anti-nausea
Anti-emetic
Serotonin (5HT3) antagonist
Dolasetron
Anti-nausea
Anti-emetic
Serotonin (5HT3) antagonist
Promethazine
Anti-nausea
Anti-emetic
Prochlorperazine
Anti-nausea
Anti-emetic
Dronabinol
Anti-nausea
Anti-emetic
Aprepitant
Anti-nausea
Anti-emetic
Loperamide
Antidiarrheal
Diphenoxylate + atropine
Lomotil
Antidiarrhea
Simethicone
Gas-X
Sulfasalazine
Anti-inflammatory
DMARD
Infliximab
Anti-inflammatory
Adalimumab
Anti-inflammatory
Methylcellulose
Bulk laxative
Psyllium
Bulk laxative
Carboxymethylcellulose
Bulk laxative
Magnesium hydroxide
Osmotic laxative
Sodium salts
Osmotic laxative
Lactulose
Osmotic laxative
Sorbitol
Osmotic laxative
Sweetener
Mannitol
Osmotic laxative
Sweetener
Polyethylene glycol
Osmotic laxative
Mineral oil
Laxative, lubricating agent
Docusate sodium
Laxative, lubricating agent
Glycerin suppositories
Laxative, lubricating agent
Lubiprostone
Prostaglandin E1 derivative
Used to treat constipation
Linaclotide
indirectly activates CFTR (increased Cl- secretion)
Used to treat constipation
Castor oil
Laxative, lubricating agent
Diphenhydramine
Very sedating first generation H1 antagonist
Dimenhydrinate
Very sedating first generation H1 antagonist
Doxylamine
Very sedating first generation H1 antagonist
Promethazine
Very sedating first generation H1 antagonist
Hydroxyzine
Very sedating first generation H1 antagonist
Brompheniramine maleate
Moderately sedating first generation H1 antagonist
Chlorpheniramine maleate
Moderately sedating first generation H1 antagonist
Clemastine
Moderately sedating first generation H1 antagonist
Cyclizine
Moderately sedating first generation H1 antagonist
Meclizine
Moderately sedating first generation H1 antagonist
Loratadine
Second generation H1 antagonist
Desloratadine
Second generation H1 antagonist
Cetirizine
Second generation H1 antagonist
Levocetirizine
Second generation H1 antagonist
Acrivistine/Pseudoephedrine
Second generation H1 antagonist
Fexofenadine
Second generation H1 antagonist
Azelastine
Nasal H1 antagonist
Levocabastine
Nasal H1 antagonist
Albuterol
Short acting B2 agonist (SABA)
Levalabuterol
Short acting B2 agonist (SABA)
Pirbuterol
Short acting B2 agonist (SABA)
Terbutaline
Short acting B2 agonist (SABA)
Salmeterol
Long acting B2 agonist (LABA)
Salmeterol/fluticasone
Long acting B2 agonist (LABA)
+
Inhaled Corticosteroid
Formoterol
Long acting B2 agonist (LABA)
Formoterol/mometasone
Long acting B2 agonist (LABA)
+
Inhaled corticosteroid
Formoterol/budesonide
Long acting B2 agonist (LABA)
+
Inhaled corticosteroid
Vilanterol/Fluticasone
Long acting B2 agonist (LABA)
+
Inhaled corticosteroid
Fluticasone
Inhaled corticosteroid
Beclomethasone
Inhaled corticosteroid
Flunisolide
Inhaled corticosteroid
Montelukast
Leukotriene inhibitor
Zafirlukast
Leukotriene inhibitor
Zileuton
Leukotriene inhibitor
Omalizumab
IgE monoclonal antibody for asthma
Benralizumab
IL-5 monoclonal antibody for eosinophilic asthma
Cromolyn sodium
For asthma: Inhibits release of histamine from mast cells
Mepolizumab
IL-5 monoclonal antibody for eosinophilic asthma
Reslizumab
IL-5 monoclonal antibody for eosinophilic asthma
Methyl salicylate (oil of winter green)
Salicylate
Celecoxib
COX-2 inhibitor
Indomethacin
Nonspecific COX inhibitor
Sulindac
Nonspecific COX inhibitor
Aspirin
Irreversible COX 1 + 2 inhibitor
Diclofenac
Nonspecific COX inhibitor
Ketorolac
Nonspecific COX inhibitor
Ibuprofen
Nonspecific COX inhibitor
Naproxen
Nonspecific COX inhibitor
Piroxicam
Nonspecific COX inhibitor
Meloxicam
Nonspecific COX inhibitor
Arthrotec
Diclofenac + Misoprostol
Acetaminophen
Nonspecific COX inhibitor
Phenylbutazone
Very potent NSAID, not available in US due to toxicities
Aurothioglucose
DMARD
Gold salt
Auranofin
DMARD
Gold salt
Gold Sodium Thiomalate
DMARD
Gold salt
Penicillamine
DMARD
Chelating agent
Hydroxychloroquine sulfate
DMARD
Infliximab
DMARD
Anti-TNF alpha drug
Adalimumab
DMARD
Anti-TNF alpha drug
Certolizumab
DMARD
Anti-TNF alpha drug
Golimumab
DMARD
Anti-TNF alpha drug
Etanercept
DMARD
Anti-TNF alpha drug
Rituximab
DMARD
Inhibitor of B cell differentiation and T cell activation
Abatacept
DMARD
Inhibitor of B cell differentiation and T cell activation
Anakinra
DMARD
Interleukin receptor antagonist
Tocilizumab
DMARD
Interleukin receptor antagonist
Leflunomide
DMARD
Inhibitor of nucleic acid synthesis
Mycophenolate mofetil
DMARD
Inhibitor of nucleic acid synthesis
Tofacitinib
JAK inhibitor
Baricitinib
JAK inhibitor
“citinib”
JAK inhibitor
“ximab”
X=crossed=chimeric monoclonal antibody
Human + murine
“mumab”
human monoclonal antibody
“zumab”
humanized monoclonal antibody
“cept”
Fusion proteins that “block/intercept” certain pathways
NOT a monoclonal antibody
“triptans”
5HTD agonists
Sumatriptan
5HTD agonist
Rizatriptan
5HTD agonist
Naratriptan
5HTD agonist
Zolmitriptan
5HTD agonist
Eletriptan
5HTD agonist
Frovatriptan
5HTD agonist
Ergotamine
Acts on 5-HT receptors
Dihydroergotamine
Acts on 5-HT receptors
Colchicine
Alkaloid, anti-inflammatory only effect for gout
Allopurinol
Xanthine oxidase inhibitor
Febuxostat
Xanthine oxidase inhibitor
Rasburicase
Enzyme that converts uric acid to allantoin
Pegloticase
Enzyme that converts uric acid to allantoin
Lesinurad
URAT1 inhibitor