Acetylcholine Drugs Flashcards
Acetylcholine
Acetylcholine agonist
Bethanechol
Direct acetylcholine agonist
Carbachol
Direct acting acetylcholine agonist
Cevimeline
Direct acting acetylcholine agonist
Methacholine
Direct acting acetylcholine agonist
Pilocarpine
Direct acting acetylcholine agonist
Excreted mainly be kidneys, acidification of urine accelerates clearance (uncharged tertiary amine)
Varenacline (Chantix)
Direct acting nicotinic-acetylcholine agonist
Pralidoxmine
Acetylcholinesterase regenerator
Ambenonium
Acetylcholinesterase inhibitor
Donepazil
Acetylcholinesterase inhibitor
Echothiophate
Acetylcholinesterase inhibitor
Edrophonium
Acetylcholinesterase inhibitor
Galantamine
Acetylcholinesterase inhibitor
Neostigmine
Acetylcholinesterase inhibitor
Physostigmine
Acetylcholinesterase inhibitor
Pyridostigmine
Acetylcholinesterase inhibitor
Rivastigmine
Acetylcholinesterase inhibitor
Tacrine
Acetylcholinesterase inhibitor
Scopolamine
Antimuscarinic drug (motion sickness)
Atropine
Antimuscarinic (GI disorders or ophthalmology)
Dicyclomine
Antimuscarinic (GI disorders)
Glycopyrrolate
Antimuscarinic (GI disorders)
Hyoscyamine
Antimuscarinic (GI disorders)
Cyclopentolate
Antimuscarinic (used in ophthalmology)
Homatropine
Antimuscarinic (used in ophthalmology)
Tropicamide
Antimuscarinic (used in ophthalmology)
Ipratropium
Antimuscarinic (used in respiratory disorders, COPD/Asthma)
Tiotropium
Antimuscarinic (used in respiratory disorders, COPD/Asthma)
Darifenacin
Antimuscarinic (used in urinary disorders)
Fesoterodine
Antimuscarinic (used in urinary disorders)
Oxybutynin
Antimuscarinic (used in urinary disorders)
Solifenacin
Antimuscarinic (used in urinary disorders)
Tolterodine
Antimuscarinic (used in urinary disorders)
Trospium
Antimuscarinic (used in urinary disorders)
Atropine + Pralidoxime
Used in cholinergic poisoning
Benztropine
Antimuscarinic (used in movement disorders)
Biperiden
Antimuscarinic (used in movement disorders)
Orphenadrine
Antimuscarinic (used in movement disorders)
Procyclidine
Antimuscarinic (used in movement disorders)
Trihexyphenidyl
Antimuscarinic (used in movement disorders)
Mecamylamine
Ganglion blocker